Ara
Toplam kayıt 65, listelenen: 21-30
Synthesis and Biological Evaluation of Novel Bischalcone Derivatives as Carbonic Anhydrase Inhibitors
(Wiley-V C H Verlag Gmbh, 2016)
Design and synthesis of a new type of bischalcones as an alternative to natural and synthetic bischalcones are reported for the first time. Key steps involved the solvent-free Claisen-Schmidt condensation of chalcones, and ...
Pyridazinone substituted benzenesulfonamides as potent carbonic anhydrase inhibitors
(Pergamon-Elsevier Science Ltd, 2016)
A series of sulfonamide derivatives (2a-l) incorporating substituted pyridazinone moieties were investigated for the inhibition of two human cytosolic carbonic anhydrase isoforms, hCA I and hCA II. All these compounds, ...
Investigation of Inhibitory Effects of Some Sulfonamides on Acethylcholinesterase Enzyme
(Wiley-Blackwell, 2016)
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Biological Evaluation of Some Uracil Derivatives as Potent Glutathione Reductase Inhibitors
(Amer Inst Physics, 2016)
Discovery of glutathione reductase (GR) inhibitors has become very popular recently due to antimalarial and anticancer activities. In this study, GR inhibitory capacities of some uracil derivatives (UDCs) (1-4) were reported. ...
Interaction of carbonic anhydrase isozymes I, II, and IX with some pyridine and phenol hydrazinecarbothioamide derivatives
(Pergamon-Elsevier Science Ltd, 2015)
A series of hydrazinecarbothioamide derivatives incorporating ethyl, phenyl, tolyl, benzyl, and allyl moieties were prepared and tested as possible inhibitors of three members of the pH regulatory enzyme family, carbonic ...
Synthesis and carbonic anhydrase inhibitory properties of novel uracil derivatives
(Pergamon-Elsevier Science Ltd, 2015)
Carbonic anhydrase (CA) inhibitors are valuable molecules based on several therapeutic applications, including antiglaucoma activity. In the present study, inhibition of two human cytosolic carbonic anhydrase isozymes I ...